The inhibition constant (Ki) of every compound was determined from the Cheng-Prusoff equation: Ki?=?IC50/(1?+?[L]/Kd), where IC50 may be the concentration of substance that displaces the binding of radioligand by 50%, [L] may be the free of charge concentration of radioligand, and Kd may be the dissociation regular of every radioligand

The inhibition constant (Ki) of every compound was determined from the Cheng-Prusoff equation: Ki?=?IC50/(1?+?[L]/Kd), where IC50 may be the concentration…

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